Name: Ifenprodil tartrate
SKU: ALK-0068

Cat#

ALK-0068

Product Name

Ifenprodil tartrate

CAS No.

23210-58-4

Description

Ifenprodil tartrate is a typical noncompetitive NMDA receptor antagonist. Ifenprodil tartrate exerts high affinity at NR1A/NR2B receptors (IC50=0.34 μM) over 400-fold than at NR1A/NR2A receptors (IC50=146 μM). Ifenprodil tartrate inhibits GIRK (Kir3), reduces inward currents through the basal GIRK activity. Ifenprodil tartrate has the potential to be a cerebral vasodilator.

Structural Formula

Ifenprodil tartrate

MW

400.49

MF

C25H33NO8

Purity

0.9995

Appearance

Solid

Solubility

DMSO : ≥ 500 mg/mL(1248.47 mM ) H2O : 5 mg/mL(12.48 mM;Need ultrasonic)

Source

Plants >Crassulaceae > Sedum sarmentosumBunge

Storage

4℃, sealed storage, away from moisture

IC50 & Target

Topoisomerase I

Shipping

Room temperature in continental US; may vary elsewhere.

SMILES

OC(C1=CC=C(O)C=C1)C(C)N(CC2)CCC2CC3=CC=CC=C3.O=C(O)[C@H](O)[C@@H](O)C(O)=O.[1/2]

In Vitro

G protein-activated inwardly rectifying K+ channels (GIRK).

Datasheet